组胺H3受体配体研究进展

吴俊;米佳丽;周成合

中国药学杂志 ›› 2007, Vol. 42 ›› Issue (06) : 404-409.

中国药学杂志 ›› 2007, Vol. 42 ›› Issue (06) : 404-409.
综述

组胺H3受体配体研究进展

  • 吴俊;米佳丽;周成合,
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摘要

目的阐述组胺H3受体配体的研究进展。方法结合国内外文献简述组胺H3受体配体及其构效关系的发展,组胺H3受体配体的治疗应用前景以及H3受体配体发展的新方向。结果与结论选择性的H3受体激动剂及拮抗剂具有广泛的生物活性,是目前抗组胺药物研究开发中的一个新的热点领域,随着对H3受体配体研究的深入,极有希望开发出可用于临床的新药。

关键词

组胺 / H3受体 / 配体 / 激动剂 / 拮抗剂

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导出引用
吴俊;米佳丽;周成合 . 组胺H3受体配体研究进展[J]. 中国药学杂志, 2007, 42(06): 404-409

参考文献

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基金

国家人事部重点项目资助课题(2002-99);教育部留学回国人员启动资金资助课题(2004-527);重庆市科委项目资助课题(2005BB5102,2002-1985);重庆医科大学创新基金;西南大学人才引进基金(SWUB2006018)

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